The book has been designed by authors based on the prodrug synthesis including the latest development in the field of prodrug methodology. We have mentioned the recent changes and developments without compromising the basic principle. New to the book Detail about prodrug methodology Brief account of HMG CoA reductase New educational features -Novel prodrug method for Simvastatin -Data tables -Guideline for further reading This book have benefitted for all those who are students of chemistry, biochemistry, Pharmaceutical sciences, Medical sciences, biotechnology and related disciplines.