1. Molecular Pharmaceutics: An Introduction 2. Protein and Enzymes Based Formulations 3. Current and Advanced Approaches in Gene Therapy 4. Vaccine and Sera 5. Aptamers and Antisense Oligonucleotides Based Delivery 6. Monoclonal Antibodies 7. Hormonal Delivery Systems 8. Vesicular Drug Delivery Systems 9. Polymeric Micelles Vs Micelles in Drug Delivery and Targeting 10. Nanoparticulate Drug Delivery Systems 11. Inorganic and Metal based Nanoparticles 12. Dendrimers: Promises and Challenges in Drug Delivery 13. Advances in Diagnostics 14. Fundamentals of Targeted Drug Delivery Systems 15. Toxicological, Clinical and Regulatory Aspects of Novel Drug Delivery Systems: Recent Updates