1. Introduction 2. Antimetabolites 3. Anticancer Drugs That Modulate Hormone Action 4. Anticancer strategies involving radical species 5. DNA Alkylating Agents 6. Anticancer Drugs That Interact with the DNA Minor Groove 7. Anticancer Drugs acting by DNA intercalation and topoisomerase inhibition 8. Epigenetic Therapy of Cancer 9. Anticancer Drugs Targeting Tubulin and Microtubules 10. Drugs Tacting on signaling pathways, part 1: Tirosine kinase inhibitors 11. Anticancer drugs acting on signaling pathways, part 2 12. Protein degradation-based cancer therapy 13. Cancer immunotherapy 14. Miscellaneous small-molecule and biological approaches to cancer therapy 15. Drug Targeting in Anticancer Chemotherapy 16. Drugs That Modulate Resistance to Anticancer Agents 17. Cancer Chemoprevention