1. Hydroxy azoles as carboxylic acid bioisosteres Marco Lucio Lucio Lolli 2. Cyclic sulfoxides & sulfones in drug design Alicia Regueiro-Ren 3. Thiazoles and topological control in drug design Robert Reid 4. Applications of fused pyrrolidine [3.3.0] heterocycles in drug design Nicholas A. Meanwell 5. 1,4 Disubstituted and 1,4,5 trisubstituted-1,2,3-triazoles in drug discovery and development: from the flask to the clinic Tracey Pirali 6. Conformationally restricted [3.2.2]- and [3.2.1]-3-azabicyclic diamines David P. Rotella
Nicholas A. Meanwell is at Bristol-Myers Squibb Research & Development, CT, USA
Marco L. Lolli is at University of Turin, Torino, Italy