1. What is Pharmacology? 2. How Different Tissues Process Drug Response 3. Drug-Receptor Theory 4. Pharmacological Assay Formats: Binding 5. Drug Targets and Drug-Target Molecules 6. Agonists: The Measurement of Affinity and Efficacy in Functional Assays 7. Orthosteric Drug Antagonism 8. Allosteric Modulation 9. The Optimal Design of Pharmacological Experiments 10. Pharmacokinetics 11. Safety Pharmacology 12. The Drug Discovery Process 13. Selected Pharmacological Methods